Falsodex ? estrogen and progesterone blocker

[chazk]

here us the profile inject it once a month and it stops progesterone and estrogen side effects, I have not seen it avialble for research or on suppliers list . Any one use and can give feed back


Falsodex is an estrogen receptor antagonist, which has no agonist effects at all. What it does is downregulates Estrogen Receptors (kinda like how Clen DownRegulates your beta receptors....so you get decreased effects from the stuff). Basically, it binds to the Estrogen Receptor more strongly then Tamoxifen, but still has no estrogen agonist effects.

The resultant down regulation of your Estrogen Receptors from the use of Falsodex results in decreased expression of the Progesterone Receptor as well! Tamoxifen, as we all know, can increase the sides from progesteronic drugs because of an increase in progesterone receptor expression. You can take Falsodex as both an anti-estrogen and an anti-progestin. You do not need to buy Arimidex (or similar drugs), and Bromocriptine!

Falsodex is administered via an IM injection of 250mgs once per month! And at that dose, it has have most if not all of the same estrogen lowering effects of 1mg/day of Arim or 2.5mgs per day of Letrozole, but has the added benefits of lowering progesterone receptor expression.

 

[macrophage69alpha]

its a super potent ER receptor antagonist. One would guess that it would destroy lipids, sex drive and anything else reliant on estrogen.

AI's lower PgR expression, by decreasing estrogen (having a similar effect), though not quite to the same extent.

IMHO this drug is not suitable for bodybuilding, it might be used for treatment of severe gyno when other treatments fail. Keeping in mind that if it last for a month any unpleasant sides will last for a month. the sides of near complete suppression of estrogen activity are not all that pleasant......