aromasin

[PARABOLAN]

where can i get some good info on this shit?? i tried the search engine and found a few things but were not enough...

 

[PARABOLAN]

come on somebody!!!!

 

[muscleup]

Its the newest and most powerful estrogen inhibitor and it supposedly like 95% effective were I've heard that arimidex is only about 75%effective, but I don't think it's out yet and I sure It's quite expensive

 

[Zyglamail]

Aromasin is available, just not something carried by most sources. Here is some cut and past on it.

AROMASIN Tablets for oral administration contain 25 mg of exemestane, an irreversible, steroidal aromatase inactivator. Exemestane is chemically described as 6-methylenandrosta-1,4-diene-3, 17-dione. Its molecular formula is C20H24O2.

The active ingredient is a white to slightly yellow crystalline powder with a molecular weight of 296.41. Exemestane is freely soluble in N, N-dimethylformamide, soluble in methanol, and practically insoluble in water.

Each AROMASIN Tablet contains the following inactive ingredients: mannitol, crospovidone, polysorbate 80, hydroxypropyl methylcellulose, colloidal silicon dioxide, microcrystalline cellulose, sodium starch glycolate, magnesium stearate, simethicone, polyethylene glycol 6000, sucrose, magnesium carbonate, titanium dioxide, methylparaben, and polyvinyl alcohol.

It comes in 25mg tabs with a retail price of around $200usd for 30 tabs.

Here is a tidbit you may be interested in

Buzdar A.

University of Texas MD Anderson Cancer Center, Houston 77030, USA. [email protected]

Exemestane is an orally active steroidal aromatase inhibitor that has demonstrated efficacy in the treatment of postmenopausal patients with advanced breast cancer. This compound exhibits a good tolerability and safety profile, which may result from its highly selective mechanism of action. Exemestane binds irreversibly to the aromatase enzyme causing inactivation of the enzyme. This irreversible loss of enzyme may contribute to the sustained inhibition of estrogen synthesis noted following exemestane administration. Exemestane is a potent inhibitor of aromatization reducing estrogen synthesis in vivo by greater than 97%. The recommended dose of exemestane is 25
mg once daily. Although dosages up to 600 mg/day have been tested, the maximum tolerated dose of exemestane has not been
reached in clinical study. The most frequently reported drug-related adverse events are hot flushes, nausea and fatigue, which are consistent with the estrogen-suppressive effects of the drug. Discontinuation due to adverse events is rare. Exemestane is a safe and well-tolerated alternative for the treatment of postmenopausal patients with advanced breast cancer.

 

[DrJMW]

Excellent post--nothing like the PDR for a few basic answers.

 

[Zyglamail]

Bump for para to see

 

[PARABOLAN]

thanx zyg ur the man...

 

[Athernigy]

.

 

[Zyglamail]

I posted more info than most people will ever attemtp to read in This thread here on EF.

 

[cbeaks]

Parabolan, I remember that you use to post about planning some pretty big cycles. Are you on one now or have one planned? What's it look like? - cbeaks